MBCY2

Prompt

2.7.11.10

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. IkappaB kinase.

AI Generated Sequence

500 AAs
MENLPPNQQTAGPWEMKERLGTGGFGNVYLWQNKETGEQIAIKQCRLELSQKNRERWCQEIQIMKRLNHPNVVKAKDVPEMLQNDVPLLAMEYCQGGDLRKLLNPENCGLRENAILSLLSDIGSALQYLHENRIIHRDLKPENIVLQDGEKLIHKIIDLGYAKEVDQGSLCTSFVGTLQYLAPELLEKQNYTVTVDYWSFGTMVFECITGYRPFLPNWQPVQWHEKIKSKDPKDIFVSEDLNGEVKFSTHLPQPNNLNSLLVERMEKWLQLLMTWDPQPRGGTDPDTPKPGCFKALDHILNLKVVHILNMVSGKIVHFPLTHEESLHSLQQRIEQETGIDPESQELLIETGALLDPRKAPTQCISDGMKLDGRRMDYDMVFLFDNSKTIYEGTFTPRSLQPDCVNSILQDPKKQLPIFQLRKVWGEAVHSISGLKEDYSRLFQGQRAAMMSLLRYNACLTKMKNSMASMSQQLKAKLDFFHTSIQIDLERYSEQMTYGIR

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT83.7
NLMSIM85.0
AACOMP91.8
Seqdif (SeqID)26.9 (PNJ34650.1)
Structdif (F-Target)9.1 (5ebz L)

ProtNLM

NameScore
2.7.11.100.510
I-kappa-B kinase0.351
Nuclear factor NF-kappa-B inhibitor kinase alpha0.038
Inhibitor of nuclear factor kappa-B kinase subunit alpha0.018
IkBKA0.011
IkBKB0.011
Designed by MP, using an AMD MI250 GPU