MQ242

Prompt

2.7.11.16

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. [G-protein-coupled receptor] kinase.

AI Generated Sequence

477 AAs
MKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMTYAFHTPDKLCFILDLMNGGDLHYHLSHHGVFSEKEMRFYATEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGTAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTVNVELPDSFSPELRSLLEGLLQRDVNKRLGCHGRGSAEVKEHPFFKGIDWQMVFLQKYPPPLIPPRGEVNAADAFDIGSFDEEDTKGIKLLDCDQELYKNFPLVISERWQQEVAETVYDAVNADTDKLERRKRAKNKQLGHEEDYAMGKDCIMHGMYGSMKLGNPFLTQWQKRYFYLFPNRLEWRGEGESPQNLLTMEQILSVEETQIKDKKCILFRIKGGKQFVLQCESDPEFVQWKKELTEAFTEAQRLLQRAPKFLNKPRSSVVELSKPPLQHRNSNGLQGSPL

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT82.0
NLMSIM85.0
AACOMP92.4
Seqdif (SeqID)5.3 (XP_046757265.1)
Structdif (F-Target)16.2 (4ra5 B)

ProtNLM

NameScore
2.7.11.-0.702
G protein-coupled receptor kinase0.259
ARBK1 kinase0.012
ARBK-10.004
G protein-coupled receptor kinase 10.003
ARBK10.002
Designed by MP, using an AMD MI250 GPU