MPXCN

Prompt

2.7.11.10

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. IkappaB kinase.

AI Generated Sequence

492 AAs
MERLPLLQQQTCGPWELKERLGTGGFGNVYRWNHKETDEKIAIKQCRLELSPKNKERWCLEIQIMKRLNHENVVKACDVPEEMANLHNDLPLLAMEYCQGGDLRKLLNQLPENCCGLKESAILTLLSDIGSALTYLHENRIIHRDLKPENIVLQQVEGKLIHKIIDLGYAKELDQGSLCTSFVGTLQYLAPELLEQKKYTVTVDYWSFGTMVFECITGFRPFLPNWQPVQWHAKIKQKDLKDIVVSEELNGEVRFSTHLPQPNNLNSLLLERMEKWLQLMLMWHPEQRGGTDPTYGPNCKFIALMDHILNLKLVHILNMTSKIITYPVRPDESLHSLQARIEAETGITASNQELLLETGASLDPRKPATQCLVDGQVDGRRVDWNPMVFLFDKSKVVYEGPFTSRSLPECVNYIVQDSKQNLPIFQLRKVWGEVWHYIQGLKEDYNRLFQGQRAAMLNLLRYNANLSKMKNSMVAFSQQLKAKLDFFKTSIQ

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT79.9
NLMSIM85.0
AACOMP91.6
Seqdif (SeqID)24.8 (XP_051688373.1)
Structdif (F-Target)8.9 (4kik B)

ProtNLM

NameScore
2.7.11.100.442
I-kappa-B kinase0.333
Nuclear factor NF-kappa-B inhibitor kinase alpha0.081
Inhibitor of nuclear factor kappa-B kinase subunit beta0.036
IkBKA0.028
IKKB kinase0.012
Designed by MP, using an AMD MI250 GPU