MLJXY

Prompt

2.7.11.16

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. [G-protein-coupled receptor] kinase.

AI Generated Sequence

688 AAs
MADLEAVLADVSYLMAMEKSKSTPAARASKKIVLPEPSIRSVMQKYLEDRGEVTFDKIFNQKIGFLLFKDYFLNEIDEAVPQLKFYEEIKEYEKLDNEEERLGRSRQIFDTYIMKELLSCSHPFSKQAVEHVQSHLAKKQVPPTLFQPYIEEICDNLRGDIFQKFMESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMTYAFHLPDKLSFILDLMNGGDLHYHLSQHGVFSEKEMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHSYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMNVELPDSFSPELKSLLEGLLQRDVSKRLGCMGRGAQEVKEHPFFKGIDWQQVFLQKYPPPLIPPRGEVNAADAFDIGSFDEEDTKGIKLLDSDQELYKNFPLTISERWQQEVAETVFDAVNADTDKIEARKRAKNKQLGHEEDYALGKDCIMHGYMLKLGNPFLTQWQRRYFYLFPNRLEWRGEGESRQNLLTMEEIVSVEETQIKDRKCILLRINGGKQFVLQCESDPEFVQWKKELTDAYREAQRLLERVPKMINKPRSPVVELSKVPLSHRSNNGL

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT82.4
NLMSIM70.0
AACOMP92.7
Seqdif (SeqID)6.0 (XP_030316745.1)
Structdif (F-Target)11.5 (4yhj A)

ProtNLM

NameScore
ARBK2 kinase0.648
ARBK1 kinase0.176
2.7.11.-0.096
G protein-coupled receptor kinase0.066
2.7.11.150.002
G protein-coupled receptor kinase 20.001
Designed by MP, using an AMD MI250 GPU