MJXS1

Prompt

2.7.11.21

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. polo kinase.

AI Generated Sequence

670 AAs
MAFANFRKIFKLGSEKKRKQYEHVKRDLNPEEVWDIIGELGDGAFGKVYKAQNKETKVLAAAKVIDTKSEEELEDYMVEIDILASCDHPNIVKLLDAFYYENNLWILIEFCAGGAVDAVMLELERPLTEPQIKVVCRQTLDALNYLHENKIIHRDLKAGNILFTLDGDIKLADFGVSAKNTRTIQRRDSFIGTPYWMAPEVVMCETSKDRPYDYKADIWSLGITLIEMAQIEPPHHEMNPMRVLLKIAKSDPPTLAQPSKWSSDFKDFLKKCLDKNVDARWTTTQLLQHPFVTVDTNKPIRELIAEAKAEVTEEVEDGKEDEEEEETENSLQIPADKRASSDLSIASSEEDKLSQNACILESLSEKTERNATGEKFSNKILNEKDTTDEPKDVVDGIHDMTNNPLEALEALDQRTAVAAEKRETEREREKPRFQPDLTDHQEQETDHINSVSKEKENTIVHTDKDKETEREDEQERFLRRQELRELRLLQKEEQRAQQQLSNKLQQQREQIFRRFEQEMTSKKRQYDQEIENLEKQQKHIEKLQKQTIERLEQEHTNRLRDEAKRIKAEQEKELSKFQNMLKENRKEVKKQQEELEKKQQELKKQQEEQKKQQEELEKQKQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQQ

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT79.5
NLMSIM70.0
AACOMP84.5
Seqdif (SeqID)17.3 (AAH47762.1)
Structdif (F-Target)2.6 (4usd A)

ProtNLM

NameScore
2.7.11.10.564
Non-specific serine/threonine protein kinase0.359
SLK kinase0.053
STK10 kinase0.003
STE20 like kinase0.002
Serine/threonine-protein kinase 100.002
Designed by MP, using an AMD MI250 GPU