MFKPX

Prompt

2.7.11.16

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. [G-protein-coupled receptor] kinase.

AI Generated Sequence

689 AAs
MADLEAVLAAVSYLMAMEKSKATPAARASKKIILPEPSIRSVMQKYLEDRGELTFDKIFNQKIGYLLFKDFCMNEIDEAVPQLKFYEEIKEYEKLDSEEERLSRSRQIYDTYIMKELLSCSHPFSKHATDHVQSHLSKKQVPPTLFQPYIEEICDSLRGGIFQKFIESDKFTRFCQWKNVELNIHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMSYAFHTPDKLSFILDLMNGGDLHYHLSQHGVFSEAEMRFYAAEIILGLEHMHNRFVVYRDLKPANILLDEFGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGVAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTMNVELPDSFSPELKSLLEGLLQRDVNKRLGCMGRGAQEVKEHPFFKGLDWQMVYLQKYPPPLIPPRGEVNAADAFDIGSFDEEDTKGIKLLDSDQELYRNFPLTISERWQQEVAETVFDAVNADTDKIEARKRAKNKQLGHEEDYALGKDCIMHGYMLKLGNPFLTQWQRRYFYLFPNRLEWRGEGESPQNLLTMEEIVSVEETQIKDKKCILLRIRGGKQFVLQCESDPELVQWKKELTEAYTEAQRLLRRAPKFLNKSRSAVVELSKVPLIHRNSTNGL

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT81.9
NLMSIM60.0
AACOMP93.2
Seqdif (SeqID)5.5 (NWY73891.1)
Structdif (F-Target)9.3 (4l9i A)

ProtNLM

NameScore
ARBK1 kinase0.348
2.7.11.-0.248
ARBK2 kinase0.205
G protein-coupled receptor kinase0.167
2.7.11.150.004
G protein-coupled receptor kinase 10.002
Designed by MP, using an AMD MI250 GPU