M3CH3

Prompt

2.7.11.16

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. [G-protein-coupled receptor] kinase.

AI Generated Sequence

685 AAs
MADLEAVLADVSYLMAMEKSKATPAARASKKIVLPEPSIRSVMQKYLEDRGEVTFDKIFNQKIGFLLFKDFAMNEIDEAVPQLKFYEEIKEYEKLDSEEERLARSREIYDTYIMKELLSCHPFSKSAVQHVSKKVQSPALFQPYIEEICQSLRGNIFQKFIESDKFTRFCQWKNVELNLHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMTYAFHTPDKLCFILDLMNGGDLHYHLSQHGVFSEKEMRFYATEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGTAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTVNVELPDSFSPELKSLLEGLLQRDVNKRLGCHGRGSQEVKEHLFFKGIDWQMVFLQKYPPPLIPPRGEVNAADAFDIGSFDEEDTKGIKLLEDCQELYKNFPLVISERWQQEVAETVFDAVNADTDKLEARKKAKNKQLGHEEDYALGKDCIMHGYMSGLKLGNPFLTKWQKRYFYLFPNRLEWRGEGESPQNLLTMEQIQSVEETQIKDKKCILFRIKGGKQFVLQCESDPEFVQWKKELTDAFTEAQRLLQRAPKFLNKPRSSVVELSKPPLQHRNSNGL

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT82.0
NLMSIM85.0
AACOMP92.5
Seqdif (SeqID)7.2 (XP_030357129.1)
Structdif (F-Target)15.4 (3nyn A)

ProtNLM

NameScore
2.7.11.-0.542
G protein-coupled receptor kinase0.307
ARBK2 kinase0.112
G protein-coupled receptor kinase 20.007
2.7.11.150.004
2.7.11.160.003
Designed by MP, using an AMD MI250 GPU