M2XAH

Prompt

2.7.11.10

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. IkappaB kinase.

AI Generated Sequence

499 AAs
MELPPVQQTCGGKWEMKERLGTGGFGNVIYRWHQLTGEQIAIKQCRLELSSKNKREWCLEIQIMKRLNHPNVVKACDVPEMEENDLPLLAMEYCSGGDLRKYLKPENCGLREQSILSLLSDISSGIQYLHEKGIIHRDLKPENIVLQEQGQLIIHKIIDLGYAKELDQGSLCTSFVGTLQYLAPELFENKPYTVTVDYWSFGTMVFECITGYRPFLHNWQPVQWSHAVKKKDKPSIFAVDEMNGEVKFSTHLPYPNNLSRLVEREMEKWLQLMLSWNPQQRGGDVLYDPKGKCFKLLDMILNLPKVHILNMMTGKVIHYSLPDETSLSQLKARIQETETGINASDQELLLETGAILDPRKTQCVADIKPWDGKGDMRYAYMVLFDKSKMTYDSSFAPRSPLDSVCNYIVQEPKLQSLPIFELRKVWGEAVHTISGLKEDYHRLFQGQRAAMSLLLRYNNALKSMKNSMSSVSQQLQAKLDFFKTSIQIDLDKYSEQTMG

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT78.9
NLMSIM85.0
AACOMP92.0
Seqdif (SeqID)34.9 (XP_023598990.1)
Structdif (F-Target)12.3 (4kik B)

ProtNLM

NameScore
2.7.11.100.502
I-kappa-B kinase0.315
Nuclear factor NF-kappa-B inhibitor kinase alpha0.074
Inhibitor of nuclear factor kappa-B kinase subunit alpha0.052
IkBKA0.014
IkBKB0.003
Designed by MP, using an AMD MI250 GPU