M2QS5

Prompt

2.7.11.15

Transferases. Transferring phosphorus-containing groups. Protein-serine/threonine kinases. [beta-adrenergic-receptor] kinase.

AI Generated Sequence

685 AAs
MADLEAVLADVSYLMAMEKSKATPAARASKKILLPEPSIRSVMQKYLEDRGEVTFDKIFNQKIGFLLFKDFAMNEIDEAVPQLKFYEEIKEYEKLDSEEERLARSREIYDTYIMKELLACHPFSKSAVQHVSKKVQSPALFQPYIEEICQSLRGNIFQKFIESDKFTRFCQWKNVELNLHLTMNDFSVHRIIGRGGFGEVYGCRKADTGKMYAMKCLDKKRIKMKQGETLALNERIMLSLVSTGDCPFIVCMTYAFHTPDKLCFILDLMNGGDLHYHLSQHGVFSEKEMRFYATEIILGLEHMHNRFVVYRDLKPANILLDEHGHVRISDLGLACDFSKKKPHASVGTHGYMAPEVLQKGTAYDSSADWFSLGCMLFKLLRGHSPFRQHKTKDKHEIDRMTLTVNVELPDSFSPELKSLLEGLLQRDVNKRLGCHGRGSQEVKEHLFFKGIDWQMVFLQKYPPPLIPPRGEVNAADAFDIGSFDEEDTKGIKLLEDCQELYKNFPLVISERWQQEVAETVFDAVNADTDKLEARKKAKNKQLGHEEDYALGKDCIMHGYMSGLKLGNPFLTKWQKRYFYLFPNRLEWRGEGESPQNLLTMEQIQSVEETQIKDKKCILFRIKGGKQFVLQCESDPEFVQWKKELTDAFTEAQRLLQRAPKFLNKPRSSVVELSKPPLQHRNSNGL

Ligand/Cofactor

ATP

C1=NC(=C2C(=N1)N(C=N2)C3C(C(C(O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N

Validation Metrics

PLDDT81.2
NLMSIM60.0
AACOMP92.5
Seqdif (SeqID)7.4 (XP_030357129.1)
Structdif (F-Target)9.3 (5uuu A)

ProtNLM

NameScore
2.7.11.-0.540
G protein-coupled receptor kinase0.302
ARBK2 kinase0.118
G protein-coupled receptor kinase 20.007
2.7.11.150.005
2.7.11.160.003
Designed by MP, using an AMD MI250 GPU